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Inner residues of macrothiolactone in autoinducer peptides I/IV circumvent spontaneous S-to-O acyl transfer to the upstream serine residue

JOURNAL ARTICLE published 2022 in RSC Chemical Biology

Research funded by Japan Society for the Promotion of Science (253534,JP16J04031,JP20H05618)

Authors: Masanobu Nagano | Satoshi Ishida | Hiroaki Suga

OligoTRAFTACs: A generalizable method for transcription factor degradation

JOURNAL ARTICLE published 2022 in RSC Chemical Biology

Research funded by National Cancer Institute (R35CA197589)

Authors: Kusal T. G. Samarasinghe | Elvira An | Miriam A. Genuth | Ling Chu | Scott A. Holley | Craig M. Crews

Understanding p300-transcription factor interactions using sequence variation and hybridization

JOURNAL ARTICLE published 2022 in RSC Chemical Biology

Research funded by Engineering and Physical Sciences Research Council (EP/N013573/1,EP/K039202/1) | Biotechnology and Biological Sciences Research Council (BB/L01386X/1) | H2020 Marie Skłodowska-Curie Actions (MSCA-IF-2016-749012) | National Research, Development and Innovation Office (NKFIH PD 135324)

Authors: Fruzsina Hóbor | Zsófia Hegedüs | Amaurys Avila Ibarra | Vencel L. Petrovicz | Gail J. Bartlett | Richard B. Sessions | Andrew J. Wilson | Thomas A. Edwards

Protein–protein interfaces in molecular glue-induced ternary complexes: classification, characterization, and prediction

JOURNAL ARTICLE published 2023 in RSC Chemical Biology

Authors: Huan Rui | Kate S. Ashton | Jaeki Min | Connie Wang | Patrick Ryan Potts

Accessing three-branched high-affinity cereblon ligands for molecular glue and protein degrader design

JOURNAL ARTICLE published 2023 in RSC Chemical Biology

Research funded by Javna Agencija za Raziskovalno Dejavnost RS (J1-2485,P1-0208) | Deutsche Forschungsgemeinschaft (Kr-3886/2-1,SFB-1074)

Authors: Robert Kuchta | Christopher Heim | Alexander Herrmann | Samuel Maiwald | Yuen Lam Dora Ng | Izidor Sosič | Tim Keuler | Jan Krönke | Michael Gütschow | Marcus D. Hartmann | Christian Steinebach

Substrate inhibition by the blockage of product release and its control by tunnel engineering

JOURNAL ARTICLE published 2021 in RSC Chemical Biology

Research funded by European Commission (857560) | Ministerstvo Školství, Mládeže a Tělovýchovy (LM2018121,LM2018140,02.1.01/0.0/0.0/18_046/0015975,CZ.02.2.69/0.0/0.0/17_050/0008496,CZ.02.2.69/0.0/0.0/19_074/0012727)

Authors: Piia Kokkonen | Andy Beier | Stanislav Mazurenko | Jiri Damborsky | David Bednar | Zbynek Prokop

Protein scaffolds: antibody alternatives for cancer diagnosis and therapy

JOURNAL ARTICLE published 2022 in RSC Chemical Biology

Authors: Renli Luo | Hongguang Liu | Zhen Cheng

Click chemistry in the development of PROTACs

JOURNAL ARTICLE published 2024 in RSC Chemical Biology

Research funded by National Institute of Diabetes and Digestive and Kidney Diseases (R01DK119202,R01DK128823)

Authors: Ce Yang | Ravi Tripathi | Binghe Wang

Nanobodies asin vivo, non-invasive, imaging agents

JOURNAL ARTICLE published 2021 in RSC Chemical Biology

Research funded by Kreftforeningen (Project no. 198164) | National Institutes of Health (1R01CA255216-01)

Authors: Thibault J. Harmand | Ashraful Islam | Novalia Pishesha | Hidde L. Ploegh

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JOURNAL ARTICLE published 2021 in RSC Chemical Biology

Correction: Fragment-based covalent ligand discovery

JOURNAL ARTICLE published 2021 in RSC Chemical Biology

Authors: Wenchao Lu | Milka Kostic | Tinghu Zhang | Jianwei Che | Matthew P. Patricelli | Lyn H. Jones | Edward T. Chouchani | Nathanael S. Gray

Finding a vocation for validation: taking proteomics beyond association and location

JOURNAL ARTICLE published 2023 in RSC Chemical Biology

Authors: Marcus J. C. Long | Jinmin Liu | Yimon Aye

Metal transport mechanism of the cation diffusion facilitator (CDF) protein family – a structural perspective on human CDF (ZnT)-related diseases

JOURNAL ARTICLE published 2021 in RSC Chemical Biology

Research funded by Israel Science Foundation (167/16) | European Cooperation in Science and Technology (CM1306)

Authors: Shiran Barber-Zucker | Arie Moran | Raz Zarivach

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JOURNAL ARTICLE published 2020 in RSC Chemical Biology

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JOURNAL ARTICLE published 2020 in RSC Chemical Biology

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JOURNAL ARTICLE published 2020 in RSC Chemical Biology

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JOURNAL ARTICLE published 2020 in RSC Chemical Biology

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JOURNAL ARTICLE published 2023 in RSC Chemical Biology

Evaluating Riboglow-FLIM probes for RNA sensing

JOURNAL ARTICLE published 2024 in RSC Chemical Biology

Research funded by American Cancer Society (ACS IRG 17-177-23) | National Institute of General Medical Sciences (R00GM127752,R35GM150823)

Authors: Nadia Sarfraz | Luke K. Shafik | Zachary R. Stickelman | Uma Shankar | Emilia Moscoso | Esther Braselmann

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JOURNAL ARTICLE published 2023 in RSC Chemical Biology